(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide
-
Catalog numberC375140
-
PricePlease ask
-
Size2,5 mg
-
-
Chemical available in other sizesPlease inquire size and price
-
Stock availabilityPlease Inquire
-
Cas number202590-98-5
-
Chemical s molecular weight491.99
-
Chemical s main applications(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide is an orally bioavailable, inhibitor of BRD2, BRD3, and BRD4 to AcH4 and shows anti-tumor activity in vitro and in vivo tumor models.
-
Chemical s categoryAmines, Aromatics, Inhibitors, Pharmaceuticals, Intermediates & Fine Chemicals, Sulfur & Selenium Compounds
-
Other name(S)-4-(4-Chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide; OTX015
-
Chemical s formulaC25H22ClN5O2S
-
Physical propertiesNo Data Available
-
Melting temperatureNo Data Available
-
Boiling temperatureNo Data Available
-
Chemical s soluble inNo Data Available
-
Stability conditionsNo Data Available
-
StorageNo Data Available
-
Gene target
-
Gene symbolMIR1302-6, PIRC28, PIRC24, PIRC26, PIRC27, PIRC25, ADCP1
-
Short name(S)-2-(4-(4-Chlorophenyl)-2 3 9-trimethyl-6H-thieno[3 2-f][1 2 4]triazolo[4 3-a][1 4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide
-
Alternative name(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide
-
Gene info
-
Identity
-
Gene
-
Long gene namemicroRNA 1302-6
-
Synonyms gene
-
Synonyms
-
Locus
-
Discovery year2008-11-03
-
Entrez gene record
-
RefSeq identity
-
Classification
- MicroRNA MIR1302 family
Gene info
-
Identity
-
Gene
-
Long gene namepiwi-interacting RNA cluster 28
-
Locus
-
Discovery year2009-11-05
-
Entrez gene record
-
Pubmed identfication
-
Classification
- Piwi-interacting RNA clusters
Gene info
-
Identity
-
Gene
-
Long gene namepiwi-interacting RNA cluster 24
-
Locus
-
Discovery year2009-11-05
-
Entrez gene record
-
Pubmed identfication
-
Classification
- Piwi-interacting RNA clusters
Gene info
-
Identity
-
Gene
-
Long gene namepiwi-interacting RNA cluster 26
-
Locus
-
Discovery year2009-11-05
-
Entrez gene record
-
Pubmed identfication
-
Classification
- Piwi-interacting RNA clusters
Gene info
-
Identity
-
Gene
-
Long gene namepiwi-interacting RNA cluster 27
-
Locus
-
Discovery year2009-11-05
-
Entrez gene record
-
Pubmed identfication
-
Classification
- Piwi-interacting RNA clusters
Gene info
-
Identity
-
Gene
-
Long gene namepiwi-interacting RNA cluster 25
-
Locus
-
Discovery year2009-11-05
-
Entrez gene record
-
Pubmed identfication
-
Classification
- Piwi-interacting RNA clusters
Gene info
-
Identity
-
Gene
-
Long gene nameadenosine deaminase complexing protein 1
-
Locus
-
Discovery year1986-01-01
-
Entrez gene record
-
Pubmed identfication
MeSH Data
-
Name
-
ConceptScope note: Radioimmunoassay of proteins using antibody coupled to an immunosorbent.
-
Tree numbers
- E05.478.566.380.830
- E05.478.566.639.830
- E05.601.470.380.830
- E05.601.470.639.830
-
Qualifiersethics, mortality, psychology, trends, veterinary, history, classification, economics, instrumentation, methods, nursing, standards, adverse effects, statistics & numerical data