Alternate Name/Synonyms
(Z)-2-(2-((3,5-dimethyl-1H-pyrrol-2-yl)methylene)-3-methoxy-2H-pyrrol-5-yl)-1H-indole methanesulfonate
Appearance
Off-white solid
CAS Number
803712-67-6
Molecular Formula
C₂₀H₁₉N₃O
Molecular Weight
317.38
Purity
≥98%
Solubility/Reconstitution Instructions
DMSO (>80 mg/ml)
Handling
Protect from air and light
Tagline
A Bcl-2 inhibitor
PubChem CID
16681698
Description
Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
