ML161
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Catalog number2689-5
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PricePlease ask
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Size5 mg
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Alternative_name2-Bromo-N-[3-[(1-oxobutyl)amino]phenyl]benzamide
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DescriptionML161 is an allosteric Inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC₅₀ = 0.26 μM for the inhibition of platelet P-selectin expression on human platelets). Also inhibits thrombin-induced platelet activation.
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CAS Number423735-93-7
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Structure AvailableY
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Salt FormNo
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Molecular FormulaC₁₇H₁₇BrN₂O₂
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Molecular Weight361.23
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Cell PermeableYes
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Purity≥98% by HPLC
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SolubilitiesDMSO (~ 30 mg/ml) or EtOH (~ 30 mg/ml)
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HandlingProtect from air and light
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Tag LineAn allosteric Inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation
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Storage Condition-20°C
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Shipping ConditionGel pack
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Shelf Life36 months
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MDL NumberMFCD03063772
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PubChem CID1048267
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SMILESCCCC(=O)NC1=CC=CC(=C1)NC(=O)C2=CC=CC=C2Br
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InChiInChI=1S/C17H17BrN2O2/c1-2-6-16(21)19-12-7-5-8-13(11-12)20-17(22)14-9-3-4-10-15(14)18/h3-5,7-11H,2,6H2,1H3,(H,19,21)(H,20,22)
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InChi KeyDFOVLSMXPWPCFH-UHFFFAOYSA-N
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MSDS AvailableYes
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Gene target
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Short nameML161
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Alternative nameML161
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