HA 130

• Catalog number
  B1192-25
• Price
  Please ask
• Size
  25 mg

• Alternative_name
  B-[3-[[4-[[3-[(4-Fluorophenyl)methyl]-2,4-dioxo-5-thiazolidinylidene]methyl]phenoxy]methyl]phenyl]-boronic acid
• Description
  HA 130 is a potent and eversible inhibitor of autotaxin (ATX) (IC₅₀ = 28 nM). It does not affect the activity of any proteasomal protease or related enzymes. HA-130 rapidly decreases plasma lysophosphatidic acid levels in mice when given intravenously (1 nM/g).
• CAS Number
  1229652-21-4
• Structure Available
  Yes
• Salt Form
  No
• Molecular Formula
  C₂₄H₁₉BFNO₅S
• Molecular Weight
  463.29
• Cell Permeable
  Yes
• Purity
  ≥98% by HPLC
• Solubilities
  DMSO (>45 mg/ml)
• Handling
  Protect from air and light
• Tag Line
  A potent and reversible inhibitor of autotaxin (ATX)
• Storage Condition
  -20°C
• Shipping Condition
  gel pack
• Shelf Life
  36 months
• PubChem CID
  46911532
• PubChem CID Link
• SMILES
  B(C1=CC=C(C=C1)COC2=CC=C(C=C2)C=C3C(=O)N(C(=O)S3)CC4=CC=C(C=C4)F)(O)O
• InChi
  1S/C24H19BFNO5S/c26-20-9-3-17(4-10-20)14-27-23(28)22(33-24(27)29)13-16-5-11-21(12-6-16)32-15-18-1-7-19(8-2-18)25(30)31/h1-13,30-31H,14-15H2/b22-13-
• InChi Key
  VTNKMYWFWQTEHE-XKZIYDEJSA-N
• Data Sheet Link
• MSDS Available
  Yes

• Gene target
  130  
• Short name
  HA 130
• Alternative name
  HA 130

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