XAV939, Tankyrase inhibitor

  • Catalog number
    SIH-532-5MG
  • Price
    Please ask
  • Size
    5 mg
  • Stock availabilitIn Stock
    In Stock
  • CAS number
    284028-89-3
  • Description
    Tankyrase inhibitor
  • Molecular weight
    312,3 g/mol
  • Primary research fields
    Cell Signaling, Epigenetics and Nuclear Signalling
  • Other name
    3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
  • Product category
    Small Molecules
  • Product type
    Inhibitor
  • Chemical formula
    C14H11F3N2OS
  • Origin
    Synthetic
  • Purity pourcentage
    >98% (HPLC); NMR (Conforms)
  • Soluble in
    Soluble in DMSO (25 mg/ml)
  • Physical appearance
    Off white powder
  • Storage recommendations
    -20ºC
  • Shipping recommendations
    Shipped Ambient
  • Safety information
    Classification: D1B Toxic Material Causing Immediate and Serious Toxic Effects - Toxic by ingestion D2B Toxic Material Causing Other Toxic Effects Moderate eye irritant Hazard statement(s): H301 Toxic if swallowed. H319 Causes serious eye irritation. Precautionary statement(s): P301 + P310 IF SWALLOWED: Immediately call a POISON CENTER or doctor/ physician. P305 + P351 + P338 IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing.
  • PubChem number
    2726824
  • Scientific context
    XAV939 is a potent tankyrase (TNKS) inhibitor, as well as a Wnt inhibitor and beta-catenin inhibitor.
  • Release date
    30/Aug/2016
  • PubMed number
    Refer to PubMed
  • Tested applications
    To be tested
  • Tested reactivity
    To be tested
  • Representative figure legend
    Chemical structure of XAV939 (SIH-532), a Tankyrase inhibitor. CAS #: 284028-89-3. Molecular Formula: C14H11F3N2OS. Molecular Weight: 312.3 g/mol. Chemical structure of XAV939, a Tankyrase inhibitor (SIH-532). CAS # 284028-89-3. Molecular Formula: C14H11F3N2OS.
  • Warning information
    Non-hazardous
  • Country of production
    Canada
  • Total weight kg
    0.25
  • Net weight g
    0.005
  • Additional description
    Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.
  • Gene target
  • Short name
    XAV939, Tankyrase inhibitor
  • Alternative name
    XAV939, Tankyrase suppressor
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