Arginine N-methyltransferase inhibitor-1
Cell-permeable. A potent and specific protein arginine N-methyltransferase (PRMTs) inhibitor (IC₅₀ = 8.8 μM for human PRMT1 and 3.0 μM for yeast Hmt1p ). Does not compete for the AdoMet (S-adenosyl-L-methionine; SAM) binding site. Also acts as a HIV-1 RT polymerase inhibitor (IC₅₀ = 5.0 μM).
Is it cell-permeable?
≥98% by NMR
Is this a salt?
Protect from light and moisture
Maximum time for storage
DMSO or Ethanol or water
For cells, cell lines and tissues in culture till half confluency.