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EPZ011989 for cell activation

EPZ011989 for cell activation is available 2 times from Biovision labs

B1221-25 | EPZ011989 for cell activation size: 25 mg | 854.96 USD

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B1221-5 | EPZ011989 for cell activation size: 5 mg | 258.63 USD

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Description EPZ011989 is a potent EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutated EZH2. It displays 15-fold selectivity for EZH2 over EZH1 and is without effect against an array of other lysine methyltransferases. EPZ011989 demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphoma.
Peptide sequence N/A
CAS number 1598383-40-4
Molecular weight 605.82
Category Biochemicals
Other name N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl((1r,4r)-4-((2-methoxyethyl)(methyl)amino)cyclohexyl)amino)-2-methyl-5-(3-morpholinoprop-1-yn-1-yl)benzamide
Molecular formula C₃₅H₅₁N₅O₄ 
Physical appearance Off-white solid
Supplied with N/A
Is this a salt? No
Is it cell-permeable? Yes
Purification ≥98% by HPLC
Reconstitute instructions DMSO(>10 mg/ml)
Storage condition -20°C
Shipping condition gel pack
Maximum time for storage 36 months
Storage instructions Protect from air and light
Additional description For cells, cell lines and tissues in culture till half confluency.
Gene targetEPZ011989 for activation
Short name EPZ011989 for activation
Technique activation
Alternative name EPZ011989 to measure cellular activation
Tissue cell
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